Comp. |
|
|
|
|
|
|
|
|
|
|
|
|
No. |
Mol-MWa |
DonorHBb |
AcceptHBc |
QPlogPo/wd |
#rotore |
PSAf |
QPlogSg |
QPlogHERGh |
QPPCacoi |
QPP |
|
|
MDCKj
|
QPlogKhsak |
% Human |
|
|
|
|
|
|
|
|
|
|
Oral |
|
|
|
|
|
|
|
|
|
|
|
|
Absorption l
|
|
|
|
|
|
|
|
|
|
|
|
|
Compound-1 |
453.3 |
1 |
5.5 |
5.5 |
5 |
63.4 |
-7.6 |
-7.1 |
2325 |
10000 |
0.714 |
100 |
Compound-2 |
276.2 |
2 |
4.7 |
2.4 |
3 |
62.8 |
-4.1 |
-5.9 |
916.1 |
450 |
-0.03 |
94.11 |
Pazopanib |
437.5 |
3 |
8.5 |
2.7 |
6 |
115.1 |
-5.88 |
-6.2 |
124.7 |
53.3 |
0.265 |
80.6 |