Aprepitant
|
NK1
|
CINV
PONV
HIV
Hot flashes
Alcohol craving/PTSD
|
Fosaprepitant
|
NK1
|
CINV
PONV
|
Casopitant
|
NK1
|
CINV
PONV
Primary insomnia
Fibromyalgia
Overactive bladder
|
Rolapitant |
NK1 |
PONV |
Orvepitant |
NK1 |
MDD |
LY-686017
|
NK1
|
SAD
Alcohol craving
|
Vofopitant
|
NK1
|
Social phobia
Primary insomnia
PTSD
|
Vestipitant
|
NK1
|
SAD
Primary insomnia
Tinnitus/hearing loss
|
AZD-2624 |
NK1 |
Schizophrenia |
SSR-240600
|
NK1
|
Overactive bladder/urge
urinary incontinence
|
TA-5538 |
NK1 |
Overactive bladder |
Saredutant
|
NK2
|
MDD
GAD
Asthma
|
Nepadutant
|
NK2
|
IBS
Asthma
POI
|
Ibodutant |
NK2 |
IBS |
DNK-333
|
NK1/NK2
|
Asthma
IBS
|
AVE-5883 |
NK1/NK2 |
Asthma |
CS-003 |
NK1/NK2/NK3 |
Asthma |
Osanetant
|
NK3
|
Schizophrenia
Panic disorder
Depression
|
Talnetant
|
NK3
|
Schizophrenia
IBS
|
SSR-241586 |
NK2/NK3 |
Schizophrenia |