Drug molecule TK receptors Clinical condition
Aprepitant
NK1
CINV PONV HIV Hot flashes Alcohol craving/PTSD
Fosaprepitant
NK1
CINV PONV
Casopitant
NK1
CINV PONV Primary insomnia Fibromyalgia Overactive bladder
Rolapitant NK1 PONV
Orvepitant NK1 MDD
LY-686017
NK1
SAD Alcohol craving
Vofopitant
NK1
Social phobia Primary insomnia PTSD
Vestipitant
NK1
SAD Primary insomnia Tinnitus/hearing loss
AZD-2624 NK1 Schizophrenia
SSR-240600
NK1
Overactive bladder/urge urinary incontinence
TA-5538 NK1 Overactive bladder
Saredutant
NK2
MDD GAD Asthma
Nepadutant
NK2
IBS Asthma POI
Ibodutant NK2 IBS
DNK-333
NK1/NK2
Asthma IBS
AVE-5883 NK1/NK2 Asthma
CS-003 NK1/NK2/NK3 Asthma
Osanetant
NK3
Schizophrenia Panic disorder Depression
Talnetant
NK3
Schizophrenia IBS
SSR-241586 NK2/NK3 Schizophrenia